Hot Sales
| Chemical Structure | Cat. No. | Product Name | CAS No. |
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BCP35590 | GS441524 New Hot Bulk | 1191237-69-0 |
GS-441524 is an adenosine nucleotide analog antiviral, similar to [remdesivir]. This molecule was patented in 2009. In vitro studies of GS-441524 have determined it has a higher EC50 than remdesivir against a number of viruses, meaning GS-441524 is less potent. GS-441524 continues to be studied in the treatment of Feline Infectious Peritonitis Virus, a coronavirus that only infects cats.
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BCP00227 | 3,4-Diaminofurazan Hot Discount Bulk | 17220-38-1 |
3,4-Diaminofurazan is a building block used to prepare magnesium and zinc alkynylated salicylaldehyde-diamine Schiff base complexes.
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BCP20294 | APR-246 New Hot Discount | 5291-32-7 |
APR-246 restores wild-type conformation and function to mutant p53, and triggers apoptosis in tumor cells. PRIMA-1Met also targets the selenoprotein thioredoxin reductase 1 (TrxR1), a key regulator of cellular redox balance.
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BCP25281 | Temsirolimus New Hot | 162635-04-3 |
Temsirolimus (CCI-779, NSC 683864) is a specific mTOR inhibitor with IC50 of 1.76 μM in a cell-free assay.
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BCP05996 | Vortioxetine New Hot | 508233-74-7 |
Vortioxetine (Lu AA21004) is an investigational novel antidepressant with multimodal activity that functions as a 5-HT3, 5-HT7 and 5-HT1D receptor antagonist, 5-HT1B receptor partial agonist, 5-HT1A receptor agonist and inhibitor of the 5-HT transporter in vitro.
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BCP02422 | Favipiravir New Hot | 259793-96-9 |
Favipiravir, also known as T705, is a RNA-directed RNA polymerase NS5B inhibitor
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BCP07838 | Delamanid New Hot | 681492-22-8 |
Delamanid, a newer mycobacterial cell wall synthesis inhibitor, inhibits the synthesisi of mucolic acids, cruciala component of the cell wall of the Mycobacterium tuberculosis complex.
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BCP19778 | Repotrectinib New Hot | 1802220-02-5 |
TPX-0005 is a potent ALK/ROS1/TRK inhibitor, with IC50 of 5.3 nM, 1.01 nM, 1.26 nM and 1.08 nM for SRC, WT ALK, ALK G1202R and ALK L1196M, respectively.
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BCP01928 | Adavosertib New Hot Discount | 955365-80-7 |
MK-1775 is a potent and selective Wee1 kinase inhibitor with an IC50 of 5.2 nM.
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BCP20662 | LOXO-195 New Hot Discount | 2097002-61-2 |
LOXO-195 is a next-generation TRK kinase (TKI) inhibitor, with IC50s of 0.6±0.1 nM, <2.5 nM for TRKA and TRKC respectively.
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BCP07998 | Bevacizumab New Hot | 216974-75-3 |
Bevacizumab is a recombinant humanized monoclonal antibody that blocks angiogenesis by inhibiting vascular endothelial growth factor A (VEGF-A).
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BCP17475 | D-glucono-1,4-lactone New Hot | 1198-69-2 |
D-glucono-1,4-lactone is a gluconolactone derived form D-gluconic acid.
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BCP09103 | Resiquimod New Hot | 144875-48-9 |
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BCP20339 | BMS-986205 New Hot Discount | 1923833-60-6 |
BMS-986205 is a selective indoleamine 2,3-dioxygenase 1 (IDO1) inhibitor.
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BCP27641 | Cabazitaxel Hot | 183133-96-2 |
A novel semi-synthetic taxane with antitumor activity used for the treatment of castration-resistant prostate cancer. A microtubule inhibitor.
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BCP20952 | Furafylline Hot | 80288-49-9 |
Furafylline is a potent and selective inhibitor of human cytochrome P450IA2 with an IC50 of 0.07 μM.
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BCP17155 | GSK2330672 Hot Discount | 1345982-69-5 |
GSK2330672 is a highly potent, nonabsorbable ASBT(apical sodium-dependent bile acid transporter) inhibitor (hASBT IC50=42 ± 3 nM) which lowers glucose in an animal model of type 2 diabetes and shows excellent developability properties for evaluating the potential therapeutic utility of a nonabsorbable ASBT inhibitor for treatment of patients with type 2 diabetes.
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BCP20094 | Nicotinamide Riboside Chloride Hot Discount Bulk | 23111-00-4 |
Nicotinamide riboside is a pyridine-nucleoside form of vitamin B3 that functions as a precursor to nicotinamide adenine dinucleotide or NAD+.
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BCP14251 | Brivaracetam Hot Discount Bulk | 357336-20-0 |
Brivaracetam(UCB-34714) is a 4-substituted pyrrolidone butanamide as agent with significant antiepileptic activity; high affinity SV2A ligand and also shows an ability to inhibit Na+ channels.
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BCP02884 | NSC 133723 Hot Discount | 19741-14-1 |
NSC 131463 is a dihydrofolate reductase potent inhibitor with an IC50 of 1 nM.
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