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Chemical Structure Cat. No. Product Name CAS No.
TTK21 Chemical Structure
BCP37892 TTK21 709676-56-2
TTK21 is an activator of CBP/p300 histone acetyltransferase activity that activates CBP/p300 histone acetyltransferase activity in a concentration-dependent manner.
CMPD101 Chemical Structure
BCP37871 CMPD101 865608-11-3
CMPD101 is a potent, highly selective and membrane-permeable small-molecule inhibitor of GRK2/3 with IC50 of 18 nM and 5.4 nM, respectively. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCα with IC50s of 3.1 μM , 2.3 μM, 1.4 μM and 8.1 μM, respectively. CMPD101 can be used for the study of heart failure.
OUL35 Chemical Structure
BCP37863 OUL35 6336-34-1
OUL35 is a small-molecule ARTD10 inhibitor. OUL35 has been shown to rescue cells from ARTD10-induced cell death.
SW155246 Chemical Structure
BCP37840 SW155246 420092-79-1
SW155246 is an inhibitor of DNA methyltransferase 1 (DNMT1) with IC50 value of 1.2 μM, displaying 30-fold selectivity for inhibition of human DNMT1 versus human or murine DNMT3A or -3B.
4'-Bromo-resveratrol Chemical Structure
BCP37824 4'-Bromo-resveratrol 1224713-90-9
4'-Bromo-resveratrol is a potent inhibitor of the deacetylases sirtuin 1 (SIRT1) and 3 (SIRT3).
GSK9311 Chemical Structure
BCP37781 GSK9311 1923851-49-3
GSK9311, a less active analogue of GSK6853, can be used as a negative control. GSK9311 inhibits BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively.
MS-402 Chemical Structure
BCP37770 MS-402 1672684-68-2
MS402 is a BD1-selective BET BrD inhibitor with Kis of 77 nM, 718 nM, 110 nM, 200 nM, 83 nM, and 240 nM for BRD4(BD1), BRD4(BD2), BRD3(BD1), BRD3(BD2), BRD2(BD1) and BRD2(BD2), respectively. MS402 blocks Th17 cell differentiation and ameliorates colitis in mice.
BAY1238097 Chemical Structure
BCP37705 BAY1238097 1564268-08-1
BAY1238097 is a potent and selective inhibitor of BET binding to histones and has strong anti-proliferative activity in different AML (acute myeloid leukemia) and MM (multiple myeloma) models through down-regulation of c-Myc levels and its downstream transcriptome (IC50 <100 nM).
IM156 Chemical Structure
BCP37661 IM156 1422365-93-2
IM156, a metformin derivative, is a potent activator of AMPK that increases AMPK phosphorylation. IM156 blocks oxidative phosphorylation (OXPHOS) through the inhibition of complex I and increases apoptosis. IM156 ameliorates various types of fibrosis and inhibits tumors.
KDM5-IN-1 Chemical Structure
BCP37630 KDM5-IN-1 1628210-26-3
KDM5-IN-1 is a potent, selective and orally bioavailable KDM5 inhibitor.
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